About 23 results found for searched term "Glucocorticoid receptor agonist" (0.201 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M13980 | Glucocorticoid receptor agonist | GCR |
| Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. IC50 value: Target: | ||
| M2176 | Dexamethasone | Animal Modeling |
| Prednisolone F; Hexadecadrol | ||
| Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist that induces the production of phospholipase A2 inhibitory protein.It can be used to construct models of allergic conjunctivitis. | ||
| M2422 | AZD5423 | GCR |
| AZD5423 is a novel nonsteroidal glucocorticoid receptor agonist. | ||
| M2626 | Dexamethasone Sodium Phosphate | Animal Modeling |
| Dexamethasone phosphate disodium | ||
| Dexamethasone Sodium Phosphate is a glucocorticoid receptor agonist that induces the production of lipocortin, a phospholipase A2 inhibitory protein. Dexamethasone inhibits autophagy levels in damaged cells in a dose-dependent manner. It can be used to construct models of allergic conjunctivitis. | ||
| M2708 | Flumethasone | Antibiotic |
| Flumetasone | ||
| Flumethasone is a glucocorticoid receptor agonist, this complex binds to the nucleus causing a variety of genetic activation and repressions. | ||
| M4882 | AL 082D06 | GCR |
| KB-145963 | ||
| AL 082D06 is a selective non-steroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM. There was no significant binding affinity for corticosteroids, androgens, estrogens and progesterone. | ||
| M5446 | Beclometasone dipropionate | GCR |
| BDP | ||
| Beclomethasone dipropionate is the precursor active molecule of Beclometasone and an orally effective glucocorticoid receptor agonist that acts through the glucocorticoid receptor to inhibit inflammation and hyperproliferation, and may be used in asthma-related studies. | ||
| M7623 | Beclomethasone | GCR |
| Beclometasone | ||
| Beclomethasone is a glucocorticoid receptor agonist with anti-inflammatory activity. | ||
| M9125 | Z-Guggulsterone | Farnesoid X Receptor |
| Z-Guggulsterone is a mineralocorticoid, progesterone and glucocorticoid receptor antagonist (Ki values are 37, 224 and 252 nM respectively) and weak androgen receptor agonist (Ki = 315 nM). | ||
| M9739 | GW-870086 | GCR |
| GW870086X | ||
| GW-870086 is a glucocorticoid receptor agonist, with pIC50 of 10.1 in A549 cells expressing NF-κB. | ||
| M11555 | Relacorilant | GCR |
| CORT 125134 | ||
| Relacorilant is a selective, oral bioeffective glucocorticoid receptor antagonist (Ki of 7.2 nM in HepG2 TAT assay and 12,81.2 nM in rat, human and monkey glucocorticoid receptor in cell-based assay). Relacorilant can be used in studies of Cushing's syndrome. | ||
| M13979 | Fluorometholone | GCR |
| Fluorometholone, a synthetic glucocorticoid, is a glucocorticoid receptor agonist with anti-inflammatory and anti-allergic properties. Fluorometholone can be used for the research of dry eye. | ||
| M13981 | Mapracorat | GCR |
| ZK-245186; BOL-303242X | ||
| Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. | ||
| M21048 | Methylprednisolone Acetate | Others |
| NSC-19987 acetate, Medrol acetate | ||
| Methylprednisolone (NSC-19987, Medrol) acetate is a synthetic glucocorticoid receptor agonist, used to achieve prompt suppression of inflammation. Methylprednisolone activates ACE2 and reduces IL-6 levels, thus improves severe or critical COVID-19. Methylprednisolone markedly reduces autophagy and apoptosis. | ||
| M21063 | LEO 134310 | Others |
| LEO 134310 is a non-steroidal, selective glucocorticoid receptor (GR) agonist that is being studied in the first phase of plaque psoriasis.LEO 134310 has shown high affinity (EC50 of 14 nM) in GR binding assays.LEO 134310 can be used in dermatological conditions. | ||
| M21281 | BAY 1003803 | GCR |
| BAY 1003803 is a glucocorticoid receptor agonist for the study of topical psoriasis or severe atopic dermatitis. | ||
| M25573 | Methylprednisolone sodium succinate | Animal Modeling |
| Methylprednisolone sodium succinate is a glucocorticoid receptor agonist with immunosuppressive and anti-inflammatory activity that can be converted to active prednisolone in vivo, thereby activating GR-mediated gene expression. In addition, Methylprednisolone sodium succinate can be used to construct a rat model of hormonal femoral head necrosis. | ||
| M27704 | Fosdagrocorat | GCR |
| PF-04171327 | ||
| Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. | ||
| M29239 | OP-3633 | GCR |
| OP-3633 is a potent and selective steroidal glucocorticoid receptor (GR) antagonist with an IC50 of 29 nM, with inhibition of GR transcriptional activity. OP-3633 exhibits low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. | ||
| M40794 | Prednisone acetate | Animal Modeling |
| Prednisone 21-acetate | ||
| Prednisone acetate is the acetate form of Prednisone and a glucocorticoid receptor agonist with anti-inflammatory and immunomodulatory properties. It can be used to construct animal models of Kawasaki disease. | ||
| M43819 | RU 26988 | GCR |
| RU 26988 is a highly specific glucocorticoid receptor agonist. | ||
| M45204 | Mometasone Furoate Monohydrate | GCR |
| Mometasone Furoate Monohydrate is a glucocorticoid receptor agonist with anti-inflammatory and anti-allergic activity. | ||
| M50237 | ORIC-101 | GCR |
| ORIC-101 is a potent and selective glucocorticoid receptor antagonist with an EC50 value of 5.6 nM and anticancer activity. | ||
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